Synthesis of novel N-substituted 3-(aminosulfonyl)-2h-l-benzopyran-2-one derivatives and their biological activity

Synthesis of novel N-substituted 3-(aminosulfonyl)-2h-l-benzopyran-2-one derivatives and their biological activity

New N-substituted 3-(aminosulfonyl)-2H-1 -benzopyran-2-one derivatives were synthesized by the reaction of salicylic aldehydes with N-substituted ethyl 2-(aminosulfonyl)acetates in the Knoevenagel condensation conditions. The structure of obtained compounds was determined through a complete IR- and...

Ausführliche Beschreibung

Gespeichert in:

Bibliographische Detailangaben
Datum:	2009
Hauptverfasser:	Kovalenko, S.S., Silin, O.V., Kovalenko, S.M., Chernykh, V.P., Maes, L., Townson, S., Yousif, F., Fakorede, F., Bernadette, R., Nwaka, S.
Format:	Artikel
Sprache:	Ukrainian
Veröffentlicht:	Інститут органічної хімії НАН України 2009
Schriftenreihe:	Журнал органічної та фармацевтичної хімії
Online Zugang:	http://dspace.nbuv.gov.ua/handle/123456789/41800
Tags:	Tag hinzufügen Keine Tags, Fügen Sie den ersten Tag hinzu!
Назва журналу:	Digital Library of Periodicals of National Academy of Sciences of Ukraine
Zitieren:	Synthesis of novel N-substituted 3-(aminosulfonyl)-2h-l-benzopyran-2-one derivatives and their biological activity / S.S. Kovalenko, O.V. Silin, S.M. Kovalenko, V.P. Chernykh, L. Maes, S. Townson, F. Yousif, F. Fakorede, R. Bernadette, S. Nwaka // Журнал органічної та фармацевтичної хімії. — 2009. — Т. 7, вип. 4(28). — С. 17-19. — Бібліогр.: 23 назв. — англ.

Institution

Digital Library of Periodicals of National Academy of Sciences of Ukraine

Ähnliche Einträge

Synthesis and biological evaluation of novel amino-substituted derivatives of pyrido[2,3-d]pyrimidine as inhibitors of protein kinase CK2
von: Zinchenko, A.N., et al.
Veröffentlicht: (2017)

Synthesis and the antimicrobial activity 1-N-alkylated derivatives of 3-N-substituted 1N-thieno (3,2-d)pirimidine-2,4-diones
von: O. V. Tkachenko, et al.
Veröffentlicht: (2013)

Investigations of solvatochromism of 2-(3-coumaroyl)-benzopyrylium dye and its di-substituted derivatives
von: Sanin, E.V., et al.
Veröffentlicht: (2013)

The synthesis of novel spirocyclic N-aryl-substituted 2-thiopyrimidine-4,6-diones
von: N. I. Kobyzhcha, et al.
Veröffentlicht: (2019)

The complexing ability of N-substituted thiourea derivatives as chelating ligands in the reaction with PdCl2
von: Yu. L. Zborovskii, et al.
Veröffentlicht: (2015)

The synthesis and the anticonvulsant activity screening of new 5-substituted 2-imino-4-thiazolidinone derivatives
von: I. A. Sydorenko, et al.
Veröffentlicht: (2022)

Synthesis and modification of 2-(coumarin-3-yl)-3,4,5,6,7,8-hexahydropyrido [4',3':4,5]thieno[2,3-d]pyrimidin-4-ones
von: Kovalenko, S.M., et al.
Veröffentlicht: (2010)

Interaction of 4-substituted 5-carbethoxy-6-chloromethylpyrimidin-2-ones with hydrazines and hydrazide derivatives: synthesis and structure
von: Lebedyeva, І.О., et al.
Veröffentlicht: (2010)

Synthesis of 1,2-benzoxathiine 2,2-dioxide derivatives using aliphatic aldehydes and assessment of their antimicrobial activity
von: G. V. Grygoriv, et al.
Veröffentlicht: (2017)

Apoptosis induction in human leukemia cells by novel 2-amino-5-benzylthiazole derivatives
von: N. S. Finiuk, et al.
Veröffentlicht: (2019)

Antineoplastic activity of novel thiazole derivatives
von: Finiuk, N.S., et al.
Veröffentlicht: (2017)

A convenient approach to the synthesis of new 4-amino substituted derivatives pyrido(2,3-d)pyrimidin-7-one
von: H. M. Zinchenko, et al.
Veröffentlicht: (2016)

The synthesis and structural functionalization of 6-substituted 2,3-dihydroimidazo
von: L. M. Saliieva, et al.
Veröffentlicht: (2018)

The efficient synthesis of 3-R-6-thio-6,7-dihydro-2H-[l,2,4]triazino[2,3-c]-quinazoline-2-ones and their derivatives, antimicrobial and antifungal activity
von: Berest, G.G., et al.
Veröffentlicht: (2010)

The plastic scintillator for n/γ-discrimination with alkyl-substituted PPO derivative.
von: Zhmurin, P.N., et al.
Veröffentlicht: (2017)

The synthesis and biological assessment of ||1,2,4|triazolo|4,3-a|pyridine-3-yl|acetamides with an 1,2,4-oxadiazol cycle in positions 6, 7 and 8
von: V. R. Karpina, et al.
Veröffentlicht: (2019)

Synthesis and alkylation of 6-(1H-benzimidazol-2-yl)-5-methylthieno |2,3-d| pyrimidin-4(3H)-ones
von: S. V. Vlasov, et al.
Veröffentlicht: (2015)

Synthesis and the antimicrobial activity of 1-alkyl-5-methyl-3-phenyl-6-(5-phenyl-1,3,4-oxadiazol-2-yl)thieno(2,3-d)pyrimidine-2,4(1H,3H)-diones
von: S. V. Vlasov, et al.
Veröffentlicht: (2015)

The study of the antimicrobial activity of the derivatives of 6-(1,2,4-oxadizol-3-yl)- and 6-(2-aminothiazol-4-yl)thieno |2,3-d| pyrimidin-4-ones by the double dilution method
von: S. V. Vlasov, et al.
Veröffentlicht: (2019)

Синтез та антимікробна активність 1-алкіл-5-метил-3-феніл-6-(5-феніл-1,3,4-оксадіазол-2-іл)тієно[2,3-d]піримідин-2,4(1H,3H)-діонів
von: Vlasov, S. V., et al.
Veröffentlicht: (2015)

Синтез та біологічна оцінка [[1,2,4]триазоло[4,3-а]піридин-3-іл]ацетамідів з 1,2,4-оксадіазольним циклом у 6, 7 та 8 положенні
von: Karpina, V. R., et al.
Veröffentlicht: (2019)

The synthesis, reactivity and the antimicrobial activity of substituted thieno(2,3-d)pyrimidine-4(3H)-thio(seleno)nes
von: D. O. Kolomieitsev, et al.
Veröffentlicht: (2015)

Синтез та алкілювання 6-(1H-бензімідазол-2-іл)-5-метилтієно[2,3-d]піримідин-4(3H)-онів
von: Vlasov, S. V., et al.
Veröffentlicht: (2015)

Regularities of isovalent atom substitution influence on the structure of AIILn2B2 IIIO7 type compounds
von: Y. A. Titov, et al.
Veröffentlicht: (2024)

Influence of intrinsic point defects and substitutional impurities (Cl, I-S) on the electronic structure of 2H-Sn2
von: D. I. Bletskan, et al.
Veröffentlicht: (2018)

Macrodialogue of Albert Camus's Novel "The Stranger"
von: V. Silin
Veröffentlicht: (2009)

Structural and dielectric properties of Ba2+ substituted lead-barium-titanate ceramics
von: P. P. Bardapurkar, et al.
Veröffentlicht: (2018)

Structural and dielectric properties of Ba2+ substituted lead-barium-titanate ceramics
von: P. P. Bardapurkar, et al.
Veröffentlicht: (2018)

Synthesis of 2-thioxo-1,2-dihydropyridine and 1,2,3,6-tetrahydropyridin-6-thione by heterocyclization of 3-amino-N-phenyl-2-butenthioamide with 2-substituted acetonitriles
von: A. N. Borisevich, et al.
Veröffentlicht: (2011)

Screening of the antiviral activity in the range of S5 and N3 substituted 4-thiazolidinone derivatives
von: D. V. Kaminskyy
Veröffentlicht: (2015)

Synthesis and antiviral activity of [(9-R1-10-R2-3-R-2-oxo-2H-[1,2,4]-triazino[2,3-s]quinazolin-6-yl)thio]acetamides derivatives with the fragments of carcass amines
von: I. S. Nosulenko, et al.
Veröffentlicht: (2014)

Crystal structure of isovalent substituted layered indates Ba1−x SrxLa2In2O7
von: Yu. O. Titov, et al.
Veröffentlicht: (2016)

The search for potential inhibitors of protein kinase Pim-1 among new amides of 1,2,4-triazolo|4,3-a|pyridine-3-metanamin with the 1,2,4-oxadiazol cycle in position 7 and 8The search for potential inhibitors of protein kinase Pim-1 among new amides of 1,2
von: V. R. Karpina, et al.
Veröffentlicht: (2019)

Enhancement of the base for 3,7-disubstituted(1,2,4)triazolo(4,3-a)pyrazin-8(7H)-one derivatives as promising pharmaceutical agents
von: Yu. Kulikovska, et al.
Veröffentlicht: (2014)

The use of aliphatic aldehydes in the synthesis of new pyran annulated derivatives of 1H-2,1-benzothiazin-4-one 2,2-dioxide via domino-type interactions. The antimicrobial activity of the compounds synthesized
von: D. A. Lega, et al.
Veröffentlicht: (2016)

Production of TlGa(In)Se2 crystals and the effect of cation substitution on their physical parameters
von: O. Parasiuk, et al.
Veröffentlicht: (2017)

Evaluation of 4H-4-chromenone derivatives as inhibitors of protein kinase CK2
von: Prykhodko, A.O., et al.
Veröffentlicht: (2005)

Novel Remote Sensing Methods for Minerals Prospecting. Chapter 2. Section 2.1-2.3
von: CASRE, SI
Veröffentlicht: (2017)

Novel Remote Sensing Methods for Minerals Prospecting. Chapter 2. Section 2.4-2.7
von: CASRE, SI
Veröffentlicht: (2017)

Novel Remote Sensing Methods for Minerals Prospecting. Chapter 2. Section 2.10-2.15
von: CASRE, SI
Veröffentlicht: (2018)